Search results for "Glycine Agents"

showing 4 items of 4 documents

Glycine receptors influence radial migration in the embryonic mouse neocortex.

2011

To investigate whether glycine receptors influence radial migration in the neocortex, we analyzed the effect of glycine and the glycinergic antagonist strychnine, on the distribution of 5-bromo-2'deoxyuridine-labeled neurons in organotypic slice cultures from embryonic mice cortices. Application of glycine impeded radial migration only in the presence of the glycine-transport blockers, ALX-5407 and ALX-1393. This effect was blocked by the specific glycine receptor antagonist strychnine, whereas application of strychnine in the absence of glycine was without effect. We conclude from these observations that an activation of glycine receptors can impede radial migration, but that the glycinerg…

GlycineCell CountNeocortexBiologychemistry.chemical_compoundMiceOrgan Culture TechniquesReceptors GlycineCell MovementGlial Fibrillary Acidic ProteinmedicineAnimalsDrug InteractionsReceptorGlycine receptorNeuronsNeocortexGeneral NeuroscienceAntagonistGlycine AgentsSarcosineGlycine receptor antagonistStrychnineStrychnineEmbryo MammalianCell biologymedicine.anatomical_structurechemistryBromodeoxyuridineCerebral cortexPhosphopyruvate HydrataseGlycineNeuroscienceNeuroreport
researchProduct

Inflammatory Pain Promotes Increased Opioid Self-Administration: Role of Dysregulated Ventral Tegmental Area μ Opioid Receptors

2015

Pain management in opioid abusers engenders ethical and practical difficulties for clinicians, often resulting in pain mismanagement. Although chronic opioid administration may alter pain states, the presence of pain itself may alter the propensity to self-administer opioids, and previous history of drug abuse comorbid with chronic pain promotes higher rates of opioid misuse. Here, we tested the hypothesis that inflammatory pain leads to increased heroin self-administration resulting from altered mu opioid receptor (MOR) regulation of mesolimbic dopamine (DA) transmission. To this end, the complete Freund's adjuvant (CFA) model of inflammation was used to assess the neurochemical and functi…

MalePain ThresholdSucroseReceptors Opioid muAction PotentialsPainMesolimbic pathwayPharmacologyHeroinRats Sprague-DawleyQuinoxalinesThreshold of painmental disordersmedicineAnimalsInflammationNeuronsGeneral NeuroscienceVentral Tegmental AreaChronic painGlycine AgentsArticlesStrychnineEnkephalin Ala(2)-MePhe(4)-Gly(5)-medicine.diseaseRatsVentral tegmental areaAnalgesics OpioidHeroinDisease Models Animalmedicine.anatomical_structureOpioidInhibitory Postsynaptic PotentialsHyperalgesiaHyperalgesiaConditioning Operantμ-opioid receptormedicine.symptomPsychologyExcitatory Amino Acid Antagonistsmedicine.drug
researchProduct

Effects of excitatory amino acids and neuropeptide Y on the discharge activity of suprachiasmatic neurons in rat brain slices

1997

Effects of L-glutamate, AMPA, NMDA and NPY on the discharge activity of neurons located in the ventral subdivision of the suprachiasmatic nucleus were examined in submerged coronal slices of the rat hypothalamus. All substances were bath applied. Application of L-glutamate (14 neurons examined) induced an excitatory response in 8 suprachiasmatic neurons (+248.9 +/- 122.24%, mean +/- S.E.M.; P0.001). A biphasic response, i.e. an initial transient excitation (+54.3 +/- 8.21%; P0.001) succeeded by an inhibition (-66.2 +/- 9.31%; P0.001), was observed in 6 neurons. Application of AMPA (36 neurons examined) resulted in an excitation of 31 neurons (+209.2 +/- 58.58%; P0.0001). Application of NMDA…

Malemedicine.medical_specialtyN-MethylaspartateGlutamic AcidAMPA receptorInhibitory postsynaptic potentialRats Sprague-Dawleychemistry.chemical_compoundOrgan Culture TechniquesInternal medicineExcitatory Amino Acid AgonistsmedicineAnimalsNeuropeptide Yalpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic AcidMolecular BiologyGlycine receptorNeuronsDose-Response Relationship DrugChemistrySuprachiasmatic nucleusGeneral NeuroscienceGlycine AgentsStrychnineStrychninehumanitiesCircadian RhythmRatsElectrophysiologyEndocrinologynervous systemHypothalamusExcitatory postsynaptic potentialNMDA receptorSuprachiasmatic NucleusNeurology (clinical)NeuroscienceDevelopmental BiologyBrain Research
researchProduct

Glycine Receptors Mediate Excitation of Subplate Neurons in Neonatal Rat Cerebral Cortex

2008

The development of the cerebral cortex depends on genetic factors and early electrical activity patterns that form immature neuronal networks. Subplate neurons (SPn) are involved in the construction of thalamocortical innervation, generation of oscillatory network activity, and in the proper formation of the cortical columnar architecture. Because glycine receptors play an important role during early corticogenesis, we analyzed the functional consequences of glycine receptor activation in visually identified SPn in neocortical slices from postnatal day 0 (P0) to P4 rats using whole cell and perforated patch-clamp recordings. In all SPn the glycinergic agonists glycine, β-alanine, and taurin…

Patch-Clamp TechniquesTaurinePhysiologyGlycineIn Vitro TechniquesBiologyMembrane PotentialsReceptors GlycineSubplatemedicineAnimalsDrug InteractionsGlycine receptorgamma-Aminobutyric AcidCerebral CortexNeuronsNeonatal ratDose-Response Relationship DrugGeneral NeuroscienceExcitatory Postsynaptic PotentialsDose-Response Relationship RadiationGlycine AgentsStrychnineElectric StimulationRatsmedicine.anatomical_structureAnimals NewbornCerebral cortexbeta-AlanineCalciumNeuroscienceJournal of Neurophysiology
researchProduct